SCHEMBL21644518

SCHEMBL21644518

CCCN(C(=O)c1cccc(F)c1)c1cc(C(C)C)c(O)cc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
HSP90AA1 P07900 5/20 0.41
HSP90AB1 P08238 1/20 0.41
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
S1PR1 P21453 2/20 0.39
MET P08581 1/20 0.39
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2B6 P20813 1/20 0.38
KMT2A Q03164 1/20 0.38
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
LMNA P02545 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30779539 1.00 TSHR (0.48) TSHRHSP90AA1HSP90AB1CES2CES1
SCHEMBL30779634 0.91 TSHR (0.59) TSHRHSP90AA1HSP90AB1CES2CES1
SCHEMBL21644643 0.91 TSHR (0.59) TSHRHSP90AA1HSP90AB1CES2CES1
SCHEMBL21644640 0.87 HSP90AA1 (0.47) HSP90AA1HSP90AB1S1PR1METCYP3A4
SCHEMBL30779618 0.87 HSP90AA1 (0.47) HSP90AA1HSP90AB1S1PR1METCYP3A4
SCHEMBL21644673 0.82 CES2 (0.44) TSHRHSP90AA1HSP90AB1CES2CES1
SCHEMBL30779585 0.82 CES2 (0.44) TSHRHSP90AA1HSP90AB1CES2CES1
SCHEMBL21644689 0.82 CES2 (0.44) TSHRHSP90AA1HSP90AB1CES2CES1
SCHEMBL30779636 0.82 CES2 (0.44) TSHRHSP90AA1HSP90AB1CES2CES1
SCHEMBL21644644 0.77 CYP3A4 (0.55) HSP90AA1METCYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111164074-B Heat shock protein 90 inhibitors 台北医学大学 2024-02-02 CN disclosed
US-11479528-B2 Heat shock protein 90 inhibitors TAIPEI MEDICAL UNIVERSITY (TW) 2022-10-25 US disclosed
CN-111164074-A Heat shock protein 90 inhibitor 台北医学大学 2020-05-15 CN disclosed
US-20200039923-A1 HEAT SHOCK PROTEIN 90 INHIBITORS TAIPEI MEDICAL UNIVERSITY (TW) 2020-02-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200039923-A1 HEAT SHOCK PROTEIN 90 INHIBITORS HSP90AB1, HSP90AB2P, HSP90AA1 TSHR 4087/4885HSP90AA1 3/4885HSP90AB1 1/4885
US-11479528-B2 Heat shock protein 90 inhibitors HSP90AB1, HSP90AB2P, HSP90AA1 TSHR 4087/4885HSP90AA1 3/4885HSP90AB1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.