SCHEMBL30779585

SCHEMBL30779585

CC(C)c1cc(N(C)C(=O)c2cccc(F)c2)c(O)cc1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
GRM1 Q13255 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRL1 P41146 1/20 0.43
TSHR P16473 3/20 0.41
HSP90AA1 P07900 6/20 0.41
CHRNB2 P17787 1/20 0.40
SLC6A2 P23975 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
SLC6A3 Q01959 1/20 0.40
HSP90AB1 P08238 1/20 0.40
PARP1 P09874 1/20 0.39
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
ADRB2 P07550 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21644673 1.00 CES2 (0.44) CES2CES1GRM1OPRM1OPRL1
SCHEMBL30779636 0.87 CES2 (0.44) CES2CES1OPRM1OPRL1TSHR
SCHEMBL21644689 0.87 CES2 (0.44) CES2CES1OPRM1OPRL1TSHR
SCHEMBL20509055 0.85 HSP90AA1 (0.43) GRM1HSP90AA1HSP90AB1HDAC1HDAC6
SCHEMBL21644643 0.84 TSHR (0.59) CES2CES1OPRM1OPRL1TSHR
SCHEMBL30779634 0.84 TSHR (0.59) CES2CES1OPRM1OPRL1TSHR
SCHEMBL30779539 0.82 TSHR (0.48) CES2CES1OPRM1OPRL1TSHR
SCHEMBL21644518 0.82 TSHR (0.48) CES2CES1OPRM1OPRL1TSHR
SCHEMBL21644586 0.74 HSP90AA1 (0.52) HSP90AA1HSP90AB1HDAC1HDAC6HDAC3
SCHEMBL21644686 0.73 POLB (0.59) HDAC1HDAC6KDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111164074-B Heat shock protein 90 inhibitors 台北医学大学 2024-02-02 CN disclosed