SCHEMBL21649219

SCHEMBL21649219

CCc1ccc2c(C(C)C)nn(C)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.41
ADORA3 P0DMS8 1/20 0.36
ADORA1 P30542 1/20 0.36
HDAC8 Q9BY41 3/20 0.36
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
MAPK8 P45983 1/20 0.33
ELANE P08246 1/20 0.33
ESR1 P03372 1/20 0.33
KIF11 P52732 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22861802 0.88 SLC22A12 (0.39) SLC22A12ADORA3ADORA1HDAC8ADORA2A
SCHEMBL21649237 0.83 SLC22A12 (0.48) SLC22A12PSEN1PSEN2APH1BNCSTN
SCHEMBL27428306 0.78 ALDH1A1 (0.41) SLC22A12ADORA3ADORA1HDAC8PSEN1
SCHEMBL18999667 0.78 ADORA2A (0.37) SLC22A12ADORA3ADORA1HDAC8ADORA2A
SCHEMBL13826298 0.78 ADORA2A (0.55) SLC22A12PSEN1PSEN2APH1BNCSTN
SCHEMBL26741066 0.78 GRM4 (0.43) SLC22A12PSEN1PSEN2APH1BNCSTN
SCHEMBL1696383 0.77 SCN9A (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL17229784 0.77 ATM (0.38) ADORA2AADORA2BMAPK8ESR1SSTR4
SCHEMBL26289032 0.77 PDGFRA (0.39) SLC22A12ADORA3ADORA1HDAC8ADORA2A
SCHEMBL21649255 0.74 ADORA2A (0.34) SLC22A12ADORA3ADORA1HDAC8ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230039309-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY 2023-02-09 US disclosed
US-11208415-B2 Substituted indole Mcl-1 inhibitors VANDERBILT UNIVERSITY (US) 2021-12-28 US disclosed
US-11160280-B2 Pesticial compounds BASF SE (DE) 2021-11-02 US disclosed
US-20210070713-A1 PESTICIDAL COMPOUNDS BASF SE (DE) 2021-03-11 US disclosed
US-20200140447-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY 2020-05-07 US disclosed
US-20200029566-A1 Pesticial Compounds BASF SE (DE) 2020-01-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200140447-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS MCL1, BCL2L1, BCL3 SLC22A12 2537/4885ADORA3 3826/4885ADORA1 3306/4885
US-11160280-B2 Pesticial compounds PNMT, DDT, NIT2 SLC22A12 1443/4885ADORA3 1873/4885ADORA1 1600/4885
US-20230039309-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS MCL1, BCL2L1, BCL3 SLC22A12 2537/4885ADORA3 3826/4885ADORA1 3306/4885
US-20210070713-A1 PESTICIDAL COMPOUNDS CAT, NIT2, PNMT SLC22A12 1787/4885ADORA3 1474/4885ADORA1 1437/4885
US-11208415-B2 Substituted indole Mcl-1 inhibitors MCL1, BCL2L1, BCL3 SLC22A12 2537/4885ADORA3 3826/4885ADORA1 3306/4885
US-20200029566-A1 Pesticial Compounds PNMT, DDT, NIT2 SLC22A12 1443/4885ADORA3 1873/4885ADORA1 1600/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.