SCHEMBL21652260

SCHEMBL21652260

CCCCc1cc(CCCC)cc(-c2ccccc2N[C@@H](c2ccccc2)[C@@H](N)c2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
FFAR4 Q5NUL3 1/20 0.34
SOAT1 P35610 2/20 0.33
KCNQ2 O43526 1/20 0.33
MAPT P10636 1/20 0.33
PSMB5 P28074 1/20 0.32
BRS3 P32247 1/20 0.31
HSD11B1 P28845 1/20 0.31
CSNK1E P49674 1/20 0.30
TACR3 P29371 1/20 0.30
DPP4 P27487 2/20 0.30
KCNH2 Q12809 1/20 0.30
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21652265 0.93 KCNQ2 (0.34) HTR2AFFAR4KCNQ2MAPTDPP4
SCHEMBL21652261 0.88 MAPT (0.36) FFAR4KCNQ2MAPTDPP4KCNH2
SCHEMBL21652277 0.81 SLC10A1 (0.41) HTR2AFFAR4BRS3
SCHEMBL21652180 0.78 DPP4 (0.36) FFAR4KCNQ2MAPTDPP4
SCHEMBL21652264 0.78 DPP4 (0.38) FFAR4KCNQ2MAPTDPP4AOC3
SCHEMBL21652160 0.77 DPP4 (0.43) KCNQ2MAPTDPP4
SCHEMBL23772891 0.75 TACR1 (0.34) FFAR4KCNQ2MAPTDPP4
SCHEMBL21652184 0.75 ABL1 (0.44) FFAR4MAPTDPP4
SCHEMBL21652182 0.74 LMNA (0.41) KCNQ2MAPTDPP4
SCHEMBL21652278 0.74 SLC10A1 (0.42) FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020019911-A1 BORON NITROGEN LIGAND BASED ON CHIRAL 1,2-ETHYLENEDIAMINE BACKBONE AND PREPARATION METHOD AND USE THEREOF 中国科学院兰州化学物理研究所苏州研究院 2020-01-30 WO disclosed