SCHEMBL21652265

SCHEMBL21652265

CCCc1cc(CCC)cc(-c2ccccc2N[C@@H](c2ccccc2)[C@@H](N)c2ccccc2)c1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 1/20 0.34
MAPT P10636 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
HTR2A P28223 1/20 0.32
DPP4 P27487 2/20 0.32
AOC3 Q16853 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21652260 0.93 HTR2A (0.39) KCNQ2MAPTFFAR4HTR2ADPP4
SCHEMBL21652261 0.90 MAPT (0.36) KCNQ2MAPTFFAR4SMN1; SMN2DPP4
SCHEMBL21652180 0.80 DPP4 (0.36) KCNQ2MAPTFFAR4SMN1; SMN2DPP4
SCHEMBL21652278 0.80 SLC10A1 (0.42) FFAR4SMN1; SMN2KDM4EALDH1A1HTT
SCHEMBL21652264 0.80 DPP4 (0.38) KCNQ2MAPTFFAR4DPP4AOC3
SCHEMBL21652160 0.79 DPP4 (0.43) KCNQ2MAPTDPP4ALDH1A1HTT
SCHEMBL23772891 0.77 TACR1 (0.34) KCNQ2MAPTFFAR4DPP4ALDH1A1
SCHEMBL21652184 0.77 ABL1 (0.44) MAPTFFAR4DPP4KDM4EALDH1A1
SCHEMBL21652182 0.76 LMNA (0.41) KCNQ2MAPTSMN1; SMN2DPP4ALDH1A1
SCHEMBL21652262 0.74 TACR1 (0.42) MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020019911-A1 BORON NITROGEN LIGAND BASED ON CHIRAL 1,2-ETHYLENEDIAMINE BACKBONE AND PREPARATION METHOD AND USE THEREOF 中国科学院兰州化学物理研究所苏州研究院 2020-01-30 WO disclosed