SCHEMBL21653174

SCHEMBL21653174

Cc1c(Cl)cccc1C(=O)Nc1c[nH]c(=O)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.46
DHODH Q02127 2/20 0.45
TOP1 P11387 3/20 0.45
MT-CO2 P00403 3/20 0.45
TP53 P04637 1/20 0.44
KCNK3 O14649 2/20 0.43
KCNK9 Q9NPC2 2/20 0.43
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ACKR3 P25106 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21653087 0.73 RAB9A (0.56) NPC1RAB9A
SCHEMBL16430801 0.73 SMN1; SMN2 (0.68) PTGS2KCNK3KCNK9ACKR3
SCHEMBL18171803 0.72 DAO (0.38) NPC1RAB9A
SCHEMBL21653175 0.71 NPC1 (0.47) TP53KCNK3KCNK9NPC1RAB9A
SCHEMBL16430921 0.69 SMN1; SMN2 (0.62) DHODHTP53NPC1RAB9A
SCHEMBL10126900 0.69 TAS1R3 (0.54) PTGS2MT-CO2TAS1R3TAS1R1TAS1R2
SCHEMBL18118631 0.68 DHODH (0.67) DHODHKCNK3KCNK9NPC1RAB9A
SCHEMBL19799127 0.68 DHODH (0.68) DHODHTP53KCNK3KCNK9NPC1
SCHEMBL3455263 0.68 CYP1A2 (0.70) TP53KCNK3KCNK9NPC1RAB9A
SCHEMBL16054667 0.68 TAS1R3 (0.52) PTGS2MT-CO2TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020023657-A1 PYRIDIN-2-ONE COMPOUNDS USEFUL AS SMARCA2 ANTAGONISTS Epizyme, Inc. (US) 2020-01-30 WO disclosed