SCHEMBL21657743

SCHEMBL21657743

Cc1ccccc1-c1c[nH]c2cc([N+](=O)[O-])ccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.54
PKLR P30613 1/20 0.54
NPBWR1 P48145 1/20 0.54
CYP19A1 P11511 1/20 0.53
CLK1 P49759 2/20 0.51
CDK5 Q00535 1/20 0.48
CDK5R1 Q15078 1/20 0.48
ELANE P08246 1/20 0.46
MAPT P10636 3/20 0.44
LMNA P02545 1/20 0.44
PTPRA P18433 1/20 0.43
DAO P14920 1/20 0.43
ALDH1A1 P00352 3/20 0.42
TDP1 Q9NUW8 3/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30283891 0.85 CYP19A1 (0.49) PKMPKLRNPBWR1CYP19A1MAPT
SCHEMBL15712649 0.81 ELANE (0.62) PKMPKLRNPBWR1CYP19A1CLK1
SCHEMBL31326013 0.81 PKM (0.56) PKMPKLRNPBWR1CLK1CDK5
SCHEMBL398147 0.81 PKM (0.56) PKMPKLRNPBWR1CLK1CDK5
SCHEMBL27510748 0.80 PKM (0.54) PKMPKLRNPBWR1CLK1CDK5
SCHEMBL14565383 0.77 TSHR (0.60) NPBWR1CYP19A1CDK5CDK5R1MAPT
SCHEMBL2033426 0.77 DAO (0.55) PKMPKLRNPBWR1CLK1CDK5
SCHEMBL21630210 0.75 IMPDH2 (0.53) CLK1CDK5CDK5R1MAPTTSHR
SCHEMBL9087198 0.75 CDK4 (0.67) PKMPKLRCLK1ELANE
SCHEMBL28855265 0.74 CLK1 (0.50) PKMPKLRCLK1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020021024-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS MODULATORS OF THE ARYL HYDROCARBON RECEPTOR (AHR) PHENEX PHARMACEUTICALS AG (DE) 2020-01-30 WO disclosed