SCHEMBL21669262

SCHEMBL21669262

COC(O)c1ccc(N)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.45
TSHR P16473 4/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPK1 P28482 1/20 0.45
ESR2 Q92731 1/20 0.43
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
RECQL P46063 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NPC1 O15118 1/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203514 0.82 SLC6A2 (0.49) CYP3A4ALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL20833999 0.78 CA12 (0.36) CYP3A4TSHRALDH1A1MAPK1HSD17B10
SCHEMBL7714921 0.76 ALDH1A1 (0.40) CYP3A4TSHRALDH1A1MAPK1ESR2
SCHEMBL24516467 0.76 ALDH1A1 (0.60) CYP3A4TSHRALDH1A1MAPK1THRB
SCHEMBL23081466 0.75 GAA (0.32) CYP3A4TSHRALOX15HSD17B10NPC1
SCHEMBL20053694 0.74 ALDH1A1 (0.50) CYP3A4ALDH1A1THRBCA1CA2
SCHEMBL10333201 0.74 TSHR (0.54) CYP3A4TSHRALDH1A1MAPK1ESR2
SCHEMBL3786798 0.74 CYP3A4 (0.54) CYP3A4TSHRALDH1A1MAPK1ESR2
SCHEMBL7680719 0.74 MEN1 (0.45) CYP3A4TSHRALDH1A1MAPK1ESR2
SCHEMBL1596051 0.73 TSHR (0.58) CYP3A4TSHRALDH1A1MAPK1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3604301-A1 4-PYRIDONE COMPOUND OR SALT THEREOF, AND PHARMACEUTICAL COMPOSITION AND FORMULATION INCLUDING SAME FUJIFILM Corporation (JP) 2020-02-05 EP disclosed