SCHEMBL2169564

SCHEMBL2169564

CS(=O)(=O)c1cc(CCCNC(=O)O)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.40
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.39
EPHX2 P34913 1/20 0.38
CCR1 P32246 1/20 0.38
KCNH2 Q12809 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
GAA P10253 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2169716 0.83 CCR1 (0.47) POLBTSHRCCR1KCNH2SMN1; SMN2
SCHEMBL9954937 0.79 NR3C2 (0.38) CCR1KCNH2SMN1; SMN2NPC1RAB9A
SCHEMBL21591538 0.77 GSK3A (0.50) POLBKDM4E
Hydrochloric Acid SCHEMBL2170595 0.76 HRH1 (0.39) CCR1KCNH2CYP2D6CYP2C19
SCHEMBL3126594 0.74 ALDH1A1 (0.41) CCR1KCNH2
SCHEMBL25374953 0.74 KDM4E (0.38) POLBKDM4ETSHREPHX2HPGD
SCHEMBL2844665 0.73 KDM4E (0.54) POLBKDM4EEPHX2SMN1; SMN2HPGD
SCHEMBL1870856 0.72 CCR1 (0.40) POLBTSHRCCR1KCNH2
Hydrochloric Acid SCHEMBL2170122 0.72 LOXL2 (0.41) KDM4ETSHRSMN1; SMN2KMT2AMEN1
SCHEMBL2644511 0.71 CCR1 (0.36) KDM4ECCR1KCNH2SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-27 EP disclosed
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed