SCHEMBL21699666

SCHEMBL21699666

COc1cccc(C2CCN(CCC3CCOCC3)CC2)n1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 18/20 0.65
DRD2 P14416 18/20 0.65
DRD4 P21917 18/20 0.65
KCNH2 Q12809 6/20 0.47
GLP1R P43220 1/20 0.42
TLR9 Q9NR96 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21699658 0.86 HTR1A (0.68) HTR1ADRD2DRD4KCNH2GLP1R
SCHEMBL21662055 0.80 DRD2 (0.57) HTR1ADRD2DRD4KCNH2GLP1R
Hydrochloric Acid SCHEMBL21642954 0.79 DRD2 (0.56) HTR1ADRD2DRD4KCNH2GLP1R
SCHEMBL21662138 0.79 DRD4 (1.00) HTR1ADRD2DRD4KCNH2
SCHEMBL17001861 0.77 DRD2 (0.52) HTR1ADRD2DRD4KCNH2TLR9
SCHEMBL14861825 0.73 HTR1A (0.47) HTR1ADRD2DRD4TLR9
SCHEMBL12093559 0.73 DDB1 (0.56) HTR1ADRD2DRD4
SCHEMBL28302369 0.70 DDB1 (0.50) HTR1ADRD2DRD4
SCHEMBL29449749 0.70 DDB1 (0.50) HTR1ADRD2DRD4
SCHEMBL27939917 0.70 DDB1 (0.50) HTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3608314-A1 2,6-DISUBSTITUTED PYRIDINE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2020-02-12 EP disclosed