SCHEMBL21699997

SCHEMBL21699997

CCOC(=O)c1c(F)c(S(N)(=O)=O)cn1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA12 O43570 2/20 0.47
CA9 Q16790 2/20 0.47
CHRNA7 P36544 5/20 0.42
STS P08842 1/20 0.41
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAOA P21397 1/20 0.37
GAA P10253 2/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
BAZ2B Q9UIF8 1/20 0.37
BAZ2A Q9UIF9 1/20 0.37
CYP2C9 P11712 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17700812 0.87 KMT2A (0.39) CA1CA2CA12CA9CHRNA7
SCHEMBL21700027 0.87 MAPT (0.40) CA1CA2CA12CA9CHRNA7
SCHEMBL16236608 0.86 BAZ2B (0.40) CA1CA2CA12CA9CHRNA7
SCHEMBL22007929 0.83 CA1 (0.48) CA1CA2CA12CA9CHRNA7
SCHEMBL22008225 0.82 STS (0.43) CA1CA2CA12CA9STS
SCHEMBL16237225 0.81 LMNA (0.38) CA1CA2KMT2AMEN1LMNA
SCHEMBL16992971 0.80 POLB (0.37) KMT2ALMNAGAATSHRHSD17B10
SCHEMBL16237218 0.79 PDK1 (0.36) KMT2ALMNAGAAALOX15TSHR
SCHEMBL18261880 0.79 PDK1 (0.36) KMT2ALMNAGAAALOX15TSHR
SCHEMBL17700858 0.79 PDK1 (0.36) KMT2ALMNAGAAALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020030781-A1 TRICYCLIC INHIBITORS OF HEPATITIS B VIRUS OSPEDALE SAN RAFFAELE S.R.L. (IT) 2020-02-13 WO disclosed
EP-3608326-A1 TRICYCLIC INHIBITORS OF HEPATITIS B VIRUS IRBM S.P.A. (IT) 2020-02-12 EP disclosed