SCHEMBL2170111

SCHEMBL2170111

NC(=O)c1cc(C(F)(F)F)ccc1OC[C@@H]1CCCNC1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 11/20 0.53
SCN8A Q9UQD0 2/20 0.51
SCN10A Q9Y5Y9 2/20 0.51
SCN9A Q15858 1/20 0.46
PDPK1 O15530 1/20 0.43
RPS6KB1 P23443 1/20 0.43
CHEK2 O96017 1/20 0.43
CHEK1 O14757 1/20 0.42
PIM1 P11309 1/20 0.42
PIM2 Q9P1W9 1/20 0.42
HTR2A P28223 1/20 0.42
PARP15 Q460N3 1/20 0.41
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2169515 0.82 CNR2 (0.51) IRAK4SCN8ASCN10A
SCHEMBL2171677 0.82 CNR2 (0.51) IRAK4SCN8ASCN10A
SCHEMBL2171142 0.80 CNR2 (0.55) IRAK4SCN10AHTR2A
SCHEMBL2170542 0.79 LTA4H (0.55) IRAK4SCN8ASCN10ASCN9A
SCHEMBL2170712 0.78 CNR2 (0.51) IRAK4SCN8ASCN10ASCN9APARP15
Tert-Butyl Formate SCHEMBL27701436 0.76 HTR2A (0.41) IRAK4SCN8ASCN10ASCN9ACHEK1
SCHEMBL3477127 0.76 TSHR (0.66) IRAK4SCN10A
SCHEMBL3443791 0.75 LTA4H (0.53) CHEK2HTR2A
SCHEMBL3443522 0.75 LTA4H (0.53) CHEK2HTR2A
SCHEMBL3443675 0.75 LTA4H (0.53) CHEK2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346843-A2 SUBSTITUTED BENZAMIDES AS CANNABINOID RECEPTOR LIGANDS Abbott Laboratories (US) 2011-07-27 EP disclosed
WO-2010028338-A2 NOVEL COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2010-03-11 WO disclosed