SCHEMBL2171677

SCHEMBL2171677

NC(=O)c1cc(C(F)(F)F)ccc1OC[C@H]1CCCN1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.51
CHRNB4 P30926 2/20 0.50
CHRNA3 P32297 2/20 0.50
LTA4H P09960 1/20 0.50
IRAK4 Q9NWZ3 3/20 0.49
MAP2K1 Q02750 1/20 0.49
RAF1 P04049 1/20 0.46
SCN8A Q9UQD0 1/20 0.46
SCN10A Q9Y5Y9 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2169515 1.00 CNR2 (0.51) CNR2CHRNB4CHRNA3LTA4HIRAK4
SCHEMBL2170542 0.97 LTA4H (0.55) CNR2CHRNB4CHRNA3LTA4HIRAK4
SCHEMBL3622371 0.84 IRAK4 (0.52) CNR2IRAK4SCN8ASCN10ATSHR
SCHEMBL2170111 0.82 IRAK4 (0.53) IRAK4SCN8ASCN10A
SCHEMBL13602330 0.81 LTA4H (0.56) CNR2CHRNB4CHRNA3LTA4H
SCHEMBL10560065 0.80 LTA4H (0.55) CHRNB4CHRNA3LTA4H
SCHEMBL3477127 0.77 TSHR (0.66) CNR2IRAK4SCN10ATSHR
SCHEMBL3159343 0.76 LTA4H (0.51) CHRNB4CHRNA3LTA4H
SCHEMBL3627815 0.76 CNR2 (0.59) CNR2CHRNB4CHRNA3IRAK4MAP2K1
SCHEMBL1974220 0.76 CNR2 (0.59) CNR2CHRNB4CHRNA3IRAK4MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346843-A2 SUBSTITUTED BENZAMIDES AS CANNABINOID RECEPTOR LIGANDS Abbott Laboratories (US) 2011-07-27 EP disclosed
WO-2010028338-A2 NOVEL COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2010-03-11 WO disclosed