SCHEMBL21702097

SCHEMBL21702097

O=C(NC1CCCCC1)C(=O)[C@@H](C[C@H]1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)c1ccc2c(c1)OCCO2

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
L3MBTL1 Q9Y468 1/20 0.45
CTSL P07711 2/20 0.41
CTSB P07858 2/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
HPGD P15428 2/20 0.41
TP53 P04637 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26494427 1.00 NPC1 (0.48) NPC1RAB9AL3MBTL1CTSLCTSB
SCHEMBL23506460 0.92 NPC1 (0.46) NPC1RAB9AL3MBTL1CTSLCTSB
SCHEMBL23711151 0.90 CTSL (0.47) NPC1RAB9AL3MBTL1CTSLCTSB
SCHEMBL23506312 0.89 SMYD3 (0.42) CTSLCTSB
SCHEMBL26495046 0.88 CTSL (0.47) RAB9ACTSLCTSBHPGD
SCHEMBL23506498 0.85 CTSL (0.47) NPC1RAB9ACTSLCTSBSMN1; SMN2
SCHEMBL21702353 0.85 SMYD3 (0.41) CTSLCTSB
SCHEMBL21702104 0.82 RAB9A (0.50) NPC1RAB9AL3MBTL1SMN1; SMN2HPGD
SCHEMBL23506496 0.82 RAB9A (0.50) NPC1RAB9AL3MBTL1SMN1; SMN2HPGD
SCHEMBL23711798 0.81 CTSL (0.46) NPC1RAB9ACTSLCTSBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3835296-A1 KETOAMIDE COMPOUND AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2021-06-16 EP disclosed
WO-2020030143-A1 KETOAMIDE COMPOUND AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF 中国科学院上海药物研究所 2020-02-13 WO disclosed