SCHEMBL21703004

SCHEMBL21703004

Nc1cccn(Cc2nc3c(COc4ccc(F)cc4F)cccc3[nH]2)c1=O

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.44
DCPS Q96C86 1/20 0.44
MAPK14 Q16539 10/20 0.41
MAP4K1 Q92918 6/20 0.38
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25942598 0.87 MAP4K1 (0.43) DHFRDCPSMAPK14MAP4K1MEN1
SCHEMBL21702996 0.80 DHFR (0.43) DHFRDCPSMAPK14MEN1ALDH1A1
SCHEMBL21703333 0.80 MAP4K1 (0.43) MAPK14MAP4K1
SCHEMBL21685623 0.80 MAP4K1 (0.56) MAP4K1
SCHEMBL25942399 0.79 MAP4K1 (0.44) MAPK14MAP4K1
SCHEMBL21703001 0.79 MAP4K1 (0.42) MAP4K1
SCHEMBL31304006 0.77 DHFR (0.50) DHFRDCPSMAPK14MAP4K1MEN1
SCHEMBL21703359 0.77 MAP4K1 (0.49) MAPK14MAP4K1
SCHEMBL21703438 0.77 MAP4K1 (0.41) MAPK14MAP4K1
SCHEMBL21703008 0.76 MAP4K1 (0.40) MAP4K1MEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020033784-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS SITARI PHARMA, INC. (US) 2020-02-13 WO disclosed