SCHEMBL2170416

SCHEMBL2170416

CN(C)c1ccccc1C(=O)NC(COCc1ccccc1)C(=O)Nc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 10/20 0.62
UGCG Q16739 6/20 0.47
TAOK1 Q7L7X3 1/20 0.46
TAOK3 Q9H2K8 1/20 0.46
NPY5R Q15761 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1375264 0.85 S1PR1 (0.68) S1PR1UGCGTAOK1TAOK3
SCHEMBL2353422 0.85 S1PR1 (0.66) S1PR1UGCGTAOK1TAOK3
SCHEMBL1374116 0.85 S1PR1 (0.62) S1PR1TAOK1TAOK3
SCHEMBL15905747 0.85 S1PR1 (0.62) S1PR1UGCGTAOK1TAOK3
SCHEMBL2353153 0.84 S1PR1 (0.72) S1PR1TAOK1TAOK3
SCHEMBL1376155 0.82 S1PR1 (0.73) S1PR1TAOK1TAOK3NPY5R
SCHEMBL1374544 0.82 UGCG (0.64) S1PR1UGCG
SCHEMBL1371986 0.82 S1PR1 (0.61) S1PR1UGCGTAOK1TAOK3
SCHEMBL1372313 0.81 S1PR1 (0.66) S1PR1TAOK1TAOK3
SCHEMBL1374223 0.81 S1PR1 (0.66) S1PR1TAOK1TAOK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed
WO-2010045580-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS EXELIXIS, INC. (US) 2010-04-22 WO disclosed