SCHEMBL2353422

SCHEMBL2353422

O=C(NC(COCc1ccccc1)C(=O)Nc1ccc(Oc2ccccc2)cc1)c1ccccc1F

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 11/20 0.66
NPC1 O15118 2/20 0.48
GAA P10253 1/20 0.48
HPGD P15428 1/20 0.48
RAB9A P51151 1/20 0.48
UGCG Q16739 2/20 0.46
TLR8 Q9NR97 1/20 0.46
TAOK1 Q7L7X3 1/20 0.46
TAOK3 Q9H2K8 1/20 0.46
TDP1 Q9NUW8 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
FAAH O00519 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1374584 0.89 S1PR1 (0.59) S1PR1UGCG
SCHEMBL1375264 0.88 S1PR1 (0.68) S1PR1UGCGTAOK1TAOK3TDP1
SCHEMBL1375613 0.88 S1PR1 (0.63) S1PR1UGCGTAOK1TAOK3
SCHEMBL2353153 0.86 S1PR1 (0.72) S1PR1NPC1RAB9ATAOK1TAOK3
SCHEMBL2170416 0.85 S1PR1 (0.62) S1PR1UGCGTAOK1TAOK3
SCHEMBL15905747 0.85 S1PR1 (0.62) S1PR1GAAUGCGTAOK1TAOK3
SCHEMBL1374368 0.85 S1PR1 (0.60) S1PR1UGCGTAOK1TAOK3
SCHEMBL1373873 0.85 S1PR1 (0.65) S1PR1NPC1RAB9ATAOK1TAOK3
SCHEMBL1373878 0.85 S1PR1 (0.65) S1PR1NPC1RAB9ATAOK1TAOK3
SCHEMBL13393225 0.85 S1PR1 (0.62) S1PR1UGCGTAOK1TAOK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed