SCHEMBL21708381

SCHEMBL21708381

Cn1cc(-c2cnc3ccc(NNC(=O)CCc4ccccc4)nc3c2)cn1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 7/20 0.68
AURKB Q96GD4 6/20 0.68
NTRK1 P04629 2/20 0.68
YES1 P07947 2/20 0.68
PIM1 P11309 1/20 0.68
WNT1 P04628 4/20 0.56
GSK3B P49841 4/20 0.56
DYRK1A Q13627 4/20 0.56
ABL1 P00519 1/20 0.55
FGFR3 P22607 3/20 0.49
FGFR4 P22455 2/20 0.49
FGFR1 P11362 2/20 0.49
FGFR2 P21802 2/20 0.49
KDR P35968 1/20 0.49
MET P08581 3/20 0.49
MST1R Q04912 1/20 0.49
HDAC8 Q9BY41 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17240002 0.88 MAPK1 (0.68) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL1933387 0.81 MAPK1 (1.00) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL15884535 0.79 MAPK1 (0.67) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL1933036 0.79 MAPK1 (0.88) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL1933048 0.79 MAPK1 (1.00) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL20950383 0.79 WNT1 (0.77) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL1932302 0.76 AURKB (1.00) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL17251852 0.76 MAPK1 (0.60) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL15884456 0.74 AURKB (0.59) MAPK1AURKBNTRK1YES1PIM1
SCHEMBL20947644 0.73 DYRK1A (0.71) MAPK1AURKBNTRK1YES1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2944637-B1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM CORP (JP) 2020-02-19 EP disclosed