SCHEMBL2170910

SCHEMBL2170910

O=C(Nc1ccc(Oc2ccc(Cl)cc2)cc1)C1CCCN1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 12/20 0.53
PFKFB1 P16118 11/20 0.53
PFKFB2 O60825 10/20 0.53
ALDH1A1 P00352 2/20 0.53
LMNA P02545 1/20 0.53
SCN3A Q9NY46 2/20 0.49
SCN9A Q15858 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
PSMB8 P28062 1/20 0.48
POLB P06746 1/20 0.48
HPGD P15428 1/20 0.48
LTA4H P09960 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23373329 1.00 PFKFB3 (0.53) PFKFB3PFKFB1PFKFB2ALDH1A1LMNA
SCHEMBL23373326 0.93 PFKFB3 (0.58) PFKFB3PFKFB1PFKFB2ALDH1A1SCN3A
SCHEMBL85092 0.92 RAB9A (0.56) ALDH1A1SCN3ASCN9ANPC1RAB9A
Hydrochloric Acid SCHEMBL76439 0.90 SCN3A (0.57) ALDH1A1SCN3ASCN9ANPC1RAB9A
Hydrochloric Acid SCHEMBL76440 0.90 SCN3A (0.57) ALDH1A1SCN3ASCN9ANPC1RAB9A
SCHEMBL23373375 0.88 PFKFB3 (0.55) PFKFB3PFKFB1PFKFB2
SCHEMBL23373378 0.88 PFKFB3 (0.61) PFKFB3PFKFB1PFKFB2SCN3ASCN9A
SCHEMBL2172458 0.87 HTR2C (0.55) PFKFB3PFKFB1PFKFB2ALDH1A1SCN3A
SCHEMBL23373331 0.87 PFKFB3 (0.56) PFKFB3PFKFB1PFKFB2SCN3ASCN9A
SCHEMBL23373327 0.86 PFKFB3 (0.55) PFKFB3PFKFB1PFKFB2SCN3ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed