SCHEMBL21709210

SCHEMBL21709210

CC1(C)c2ccccc2-c2c(N(c3ccc(-c4ccccc4)cc3)c3nc(-c4ccc(-c5cccc6ccccc56)cc4)c4ccccc4n3)cccc21

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.40
SCN9A Q15858 1/20 0.33
PPARG P37231 7/20 0.32
PPARA Q07869 7/20 0.32
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PPARD Q03181 1/20 0.31
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709288 0.95 NUDT1 (0.44) NUDT1SCN9A
SCHEMBL21679716 0.95 NUDT1 (0.44) NUDT1SCN9A
SCHEMBL21709281 0.92 NUDT1 (0.42) NUDT1SCN9A
SCHEMBL21709377 0.90 NUDT1 (0.47) NUDT1SCN9A
SCHEMBL21709208 0.89 NUDT1 (0.38) NUDT1SCN9A
SCHEMBL21709418 0.89 NUDT1 (0.40) NUDT1SCN9A
SCHEMBL26002170 0.88 CA12 (0.37) PPARGPPARACYP2C9CYP2C19PPARD
SCHEMBL26002157 0.88 CA12 (0.37) PPARGPPARACYP2C9CYP2C19PPARD
SCHEMBL21709286 0.88 NUDT1 (0.36) NUDT1SCN9A
SCHEMBL21709205 0.87 NUDT1 (0.38) NUDT1SCN9ACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200048207-A1 COMPOUNDS WITH ARYLAMINE STRUCTURES MERCK PATENT GMBH (DE) 2020-02-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200048207-A1 COMPOUNDS WITH ARYLAMINE STRUCTURES DDT, NAT1, INMT NUDT1 15/4885SCN9A 1893/4885PPARG 2428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.