SCHEMBL21709653

SCHEMBL21709653

C#C[C@@]1(CO[SiH](C)C(C)(C)C)CC[C@H](n2cnc3c(N)nc(F)nc32)O1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AHCY P23526 4/20 0.40
NT5E P21589 6/20 0.38
LMNA P02545 2/20 0.38
HIF1A Q16665 1/20 0.38
CHKA P35790 3/20 0.36
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 2/20 0.35
ADORA1 P30542 2/20 0.35
CA5A P35218 1/20 0.35
ADORA2B P29275 1/20 0.35
DNMT1 P26358 1/20 0.31
DNMT3B Q9UBC3 1/20 0.31
PNP P00491 1/20 0.31
TP53 P04637 1/20 0.31
HTT P42858 1/20 0.31
PDE4D Q08499 1/20 0.31
PDE3A Q14432 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21347881 0.89 AHCY (0.35) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL25659855 0.85 AHCY (0.45) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL12214180 0.85 AHCY (0.41) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL21347920 0.83 CHKA (0.40) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL22855175 0.83 AHCY (0.47) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL2520516 0.83 AHCY (0.47) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL13581562 0.82 AHCY (0.42) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL21347509 0.82 CHKA (0.39) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL22939391 0.82 CHKA (0.44) AHCYNT5ELMNAHIF1ACHKA
SCHEMBL21347049 0.81 CHKA (0.40) AHCYNT5ELMNAHIF1ACHKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020031131-A1 COMPOUNDS USEFUL IN HIV THERAPY GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2020-02-13 WO disclosed