SCHEMBL21709998

SCHEMBL21709998

Cc1ccc(OC(C)C)c(OC(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
ACHE P22303 1/20 0.42
MEN1 O00255 9/20 0.42
KMT2A Q03164 9/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
MAPT P10636 5/20 0.42
LMNA P02545 5/20 0.42
MAPK1 P28482 2/20 0.42
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
CSNK2A1 P68400 2/20 0.39
GAA P10253 2/20 0.38
HTT P42858 2/20 0.36
ATM Q13315 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
TSHR P16473 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15521568 1.00 ALDH1A1 (0.46) ALDH1A1ACHEMEN1KMT2ASMN1; SMN2
SCHEMBL14345864 0.92 ALDH1A1 (0.51) ALDH1A1ACHEMEN1KMT2ASMN1; SMN2
SCHEMBL12313570 0.90 ACHE (0.50) ALDH1A1ACHESMN1; SMN2MAPTLMNA
SCHEMBL12180465 0.82 ACHE (0.65) ALDH1A1ACHEMEN1KMT2ASMN1; SMN2
SCHEMBL15133865 0.82 ACHE (0.65) ALDH1A1ACHEMEN1KMT2ASMN1; SMN2
SCHEMBL10196610 0.80 ACHE (0.68) ALDH1A1ACHEMEN1KMT2ASMN1; SMN2
SCHEMBL10196623 0.80 ACHE (0.68) ALDH1A1ACHEMEN1KMT2ASMN1; SMN2
SCHEMBL28651200 0.79 PDE4A (0.35) ALDH1A1SMN1; SMN2LMNAMAPK1TP53
SCHEMBL2088008 0.79 GAA (0.43) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL131996 0.79 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11192886-B2 S1P1 agonist and application thereof MEDSHINE DISCOVERY INC. (CN) 2021-12-07 US disclosed
US-20210300908-A1 S1P1 AGONIST AND APPLICATION THEREOF Shijiazhuang Sagacity New Drug Development Co., Ltd. (CN) 2021-09-30 US disclosed
US-10981900-B2 Spiro compound and use thereof MEDSHINE DISCOVERY INC. (CN) 2021-04-20 US disclosed
US-20200048235-A1 SPIRO COMPOUND AND USE THEREOF MEDSHINE DISCOVERY INC. (CN) 2020-02-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200048235-A1 SPIRO COMPOUND AND USE THEREOF S1PR1, S1PR2, S1PR3 ALDH1A1 862/4885ACHE 4560/4885MEN1 747/4885
US-11192886-B2 S1P1 agonist and application thereof S1PR1, S1PR2, S1PR3 ALDH1A1 2418/4885ACHE 4137/4885MEN1 1009/4885
US-10981900-B2 Spiro compound and use thereof S1PR1, S1PR2, S1PR3 ALDH1A1 862/4885ACHE 4560/4885MEN1 747/4885
US-20210300908-A1 S1P1 AGONIST AND APPLICATION THEREOF S1PR1, S1PR2, S1PR3 ALDH1A1 2418/4885ACHE 4137/4885MEN1 1009/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.