SCHEMBL21714966

SCHEMBL21714966

CNC(=O)C1CN=C(C2CCNCC2)C=N1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
HTR1F P30939 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA4 P43681 1/20 0.30
PLAT P00750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21712556 0.81 PARP1 (0.36) GABRA1GABRB2PLAT
SCHEMBL21715179 0.74 TSHR (0.45)
SCHEMBL21714937 0.72 CHRNB2 (0.30) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL2918633 0.64 POLB (0.36) GABRA1GABRB2CHRNB2CHRNB4CHRNA3
SCHEMBL2917663 0.62 CHRNB2 (0.36) GABRA1GABRB2CHRNB2CHRNB4CHRNA3
SCHEMBL5326 0.62 POLB (0.54) GABRA1GABRB2CHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL4788809 0.60 POLB (0.52) GABRA1GABRB2CHRNB2CHRNB4CHRNA3
SCHEMBL4179238 0.58 HDAC8 (0.51)
SCHEMBL17623531 0.57 CHRNB2 (0.31) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL2915344 0.57 PRCP (0.39) GABRA1GABRB2CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020029980-A1 SMAD3 INHIBITORS MOEXA PHARMACEUTICALS LIMITED (CN) 2020-02-13 WO disclosed