SCHEMBL21725009

SCHEMBL21725009

NC(=O)c1cn(C(N)=O)c2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 12/20 0.49
MEN1 O00255 3/20 0.49
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 3/20 0.45
THRB P10828 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
FABP4 P15090 1/20 0.44
TSHR P16473 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CREBBP Q92793 1/20 0.43
MAPT P10636 2/20 0.42
ATM Q13315 1/20 0.42
CNR1 P21554 1/20 0.42
POLB P06746 1/20 0.41
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12479862 0.87 ALDH1A1 (0.48) KMT2AMEN1KDM4EALDH1A1THRB
SCHEMBL27387445 0.87 KMT2A (0.48) KMT2AMEN1KDM4EALDH1A1THRB
SCHEMBL30394690 0.86 CREBBP (0.58) KMT2AMEN1KDM4EALDH1A1THRB
SCHEMBL8359818 0.86 KMT2A (0.60) KMT2AMEN1KDM4EALDH1A1THRB
SCHEMBL25428769 0.83 LMNA (0.50) KMT2AMEN1KDM4EALDH1A1THRB
SCHEMBL4205321 0.82 KMT2A (0.47) KMT2AMEN1KDM4EALDH1A1THRB
SCHEMBL10596904 0.81 KDM4E (0.50) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL19668173 0.80 LMNA (0.56) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL12481379 0.79 KDM4E (0.41) KMT2AMEN1KDM4EALDH1A1THRB
SCHEMBL8530588 0.79 KDM4E (0.41) KMT2AMEN1KDM4EALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111303148-B 1-substituted beta-carboline derivatives and application thereof 南京农业大学 2022-08-30 CN disclosed
WO-2020037116-A1 SMALL MOLECULE PYRIN-DOMAIN TARGETED NLRP3 INFLAMMASOME INHIBITORS H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2020-02-20 WO disclosed