SCHEMBL21732265

SCHEMBL21732265

CC(=O)N1Cc2cc([S+](C)[O-])ccc2C1C(=O)Nc1cnc(N2CCCC2c2cccc(C(F)(F)F)c2)nc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 18/20 0.41
CYP2D6 P10635 12/20 0.41
IL17A Q16552 1/20 0.40
KCNH2 Q12809 4/20 0.40
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21732120 0.93 RORC (0.43) RORCCYP2D6IL17AKCNH2
SCHEMBL21732119 0.91 NTRK1 (0.41)
SCHEMBL21732214 0.90 RORC (0.36) RORCCYP2D6IL17AKCNH2
SCHEMBL21732208 0.89 RORC (0.39) RORCCYP2D6IL17AKCNH2
SCHEMBL21732266 0.88 RORC (0.38) RORCCYP2D6IL17AKCNH2
SCHEMBL21732188 0.88 RORC (0.38) RORCCYP2D6IL17AKCNH2
SCHEMBL21732206 0.86 RORC (0.37) RORCCYP2D6IL17AKCNH2
SCHEMBL21732254 0.84 NTRK1 (0.41)
SCHEMBL21732221 0.83 RORC (0.42) RORCCYP2D6IL17AKCNH2
SCHEMBL21732220 0.82 NTRK1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035557-A1 NOVEL HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2020-02-20 WO disclosed