SCHEMBL21733955

SCHEMBL21733955

N=C(OC(=N)C1CC1)C1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 4/20 0.46
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MGLL Q99685 1/20 0.36
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
EPHX1 P07099 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21733958 0.85 NOS2 (0.39) NOS2CES2CES1MGLLHDAC8
SCHEMBL909692 0.78 NOS2 (0.42) NOS2CES2CES1MGLLHDAC8
Hydrochloric Acid SCHEMBL4532413 0.76 NOS2 (0.40) NOS2CES2CES1MGLLHDAC8
SCHEMBL24043609 0.73 NOS2 (0.48) NOS2CES2CES1MGLLHDAC8
SCHEMBL8166352 0.73
SCHEMBL18800430 0.73 NOS2 (0.48) NOS2CES2CES1MGLLHDAC8
SCHEMBL507070 0.72 ALDH1A1 (0.46) NOS2CES2CES1ALDH1A1TSHR
Hydrochloric Acid SCHEMBL20819822 0.72 NOS2 (0.42) NOS2CES2CES1HDAC8HDAC6
SCHEMBL879167 0.71 NOS2 (0.53) NOS2CES2CES1MGLLHDAC8
Hydrochloric Acid SCHEMBL506728 0.71 ALDH1A1 (0.44) NOS2CES2CES1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020036979-A1 PYRROLO[1,2-B]PYRIDAZINE DERIVATIVES AS IRAK4 INHIBITORS GILEAD SCIENCES, INC. (US) 2020-02-20 WO disclosed