SCHEMBL21734020

SCHEMBL21734020

Cc1ccc2cnn(PI)c2c1C1CCc2c(nc[nH]c2=O)C1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 1/20 0.33
KRAS P01116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24854593 0.85 GRM7 (0.43) GRM7KRAS
SCHEMBL21733780 0.80 CYP4F2 (0.35) GRM7
SCHEMBL30834498 0.80 CYP4F2 (0.35) GRM7
SCHEMBL21734021 0.78 KRAS (0.38) GRM7KRAS
SCHEMBL21734019 0.77 MAPT (0.33)
SCHEMBL21733818 0.73 KRAS (0.51) KRAS
SCHEMBL30834503 0.72 GRM7 (0.32) GRM7KRAS
SCHEMBL21722189 0.72 GRM7 (0.32) GRM7KRAS
SCHEMBL21733500 0.70 KRAS (0.36) GRM7KRAS
SCHEMBL21733527 0.70 MEN1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11760744-B2 Fused ring compounds GENENTECH, INC. (US) 2023-09-19 US disclosed
US-20230002345-A1 FUSED RING COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2023-01-05 US disclosed
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11760744-B2 Fused ring compounds KRAS, NRAS, HRAS GRM7 2937/4885KRAS 1/4885
US-20230002345-A1 FUSED RING COMPOUNDS KRAS, NRAS, HRAS GRM7 2937/4885KRAS 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.