SCHEMBL21722189

SCHEMBL21722189

Cc1ccc2c(c1C1CCc3c(nc[nH]c3=O)C1)COC2

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 1/20 0.32
KRAS P01116 1/20 0.32
SRC P12931 2/20 0.31
ADRA1A P35348 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30834503 1.00 GRM7 (0.32) GRM7KRASSRCADRA1A
SCHEMBL21734011 0.73 KRAS (0.41) GRM7KRAS
SCHEMBL21722231 0.73 KRAS (0.41) GRM7KRAS
SCHEMBL30834506 0.73 KRAS (0.41) GRM7KRAS
SCHEMBL20836477 0.72 GRM7 (0.46) GRM7ADRA1A
SCHEMBL31483708 0.72 GRM7 (0.46) GRM7ADRA1A
SCHEMBL21722290 0.72 MAPT (0.36)
SCHEMBL21733758 0.72 KMT2A (0.39)
SCHEMBL24854593 0.72 GRM7 (0.43) GRM7KRAS
SCHEMBL21734020 0.72 GRM7 (0.33) GRM7KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11760744-B2 Fused ring compounds GENENTECH, INC. (US) 2023-09-19 US disclosed
US-11760744-B2 Fused ring compounds GENENTECH, INC. (US) 2023-09-19 US disclosed
US-20230002345-A1 FUSED RING COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2023-01-05 US disclosed
EP-3746436-A1 FUSED RING COMPOUNDS F. Hoffmann-La Roche AG (CH) 2020-12-09 EP disclosed
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11760744-B2 Fused ring compounds KRAS, NRAS, HRAS GRM7 2937/4885KRAS 1/4885SRC 551/4885
US-20230002345-A1 FUSED RING COMPOUNDS KRAS, NRAS, HRAS GRM7 2937/4885KRAS 1/4885SRC 551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.