SCHEMBL21739715

SCHEMBL21739715

Cc1cccc2c1NC(C(=O)N[C@H]1CC[C@H](C(F)(F)F)CC1)C2

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.39
PTGES O14684 1/20 0.36
DRD2 P14416 2/20 0.36
HTR2A P28223 1/20 0.36
DRD3 P35462 1/20 0.36
EPHX1 P07099 1/20 0.34
RAB9A P51151 2/20 0.33
KMT2A Q03164 1/20 0.33
EPHX2 P34913 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21740209 0.89 SMYD3 (0.39) SMYD3DRD2HTR2ADRD3EPHX1
SCHEMBL21739907 0.86 SMYD3 (0.42) SMYD3EPHX1RAB9AKMT2AEPHX2
SCHEMBL21740213 0.86 MTNR1A (0.44) SMYD3DRD2EPHX1RAB9AKMT2A
SCHEMBL21739921 0.84 EPHX1 (0.49) EPHX1RAB9AKMT2AEPHX2NPC1
SCHEMBL21739422 0.84 PTGES (0.42) SMYD3PTGESDRD2EPHX1KMT2A
SCHEMBL21739169 0.83 POLB (0.41) SMYD3HTR2AEPHX1RAB9AKMT2A
SCHEMBL25040289 0.82 SSTR4 (0.42) SMYD3RAB9AKMT2AEPHX2ALDH1A1
SCHEMBL21739908 0.82 SMYD3 (0.39) SMYD3PTGESEPHX1RAB9AKMT2A
SCHEMBL21740347 0.81 SMYD3 (0.50) SMYD3
SCHEMBL22052079 0.80 KMT2A (0.42) SMYD3EPHX1RAB9AKMT2AEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020112872-A1 METHODS OF TREATING WHSC1-OVEREXPRESSING CANCERS BY INHIBITING SETD2 Epizyme, Inc. (US) 2020-06-04 WO disclosed
WO-2020037079-A1 SUBSTITUTED INDOLES AND METHODS OF USE THEREOF Epizyme, Inc. (US) 2020-02-20 WO disclosed