SCHEMBL21742813

SCHEMBL21742813

CNCCCc1cnco1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
NAMPT P43490 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373758 0.78
SCHEMBL460224 0.76 CYP3A4 (0.41) ALDH1A1MAPTHRH4HRH3L3MBTL1
SCHEMBL13949575 0.75
SCHEMBL21210714 0.74 CYP3A4 (0.40) MEN1KMT2AALDH1A1MAPTL3MBTL1
SCHEMBL5544928 0.74
SCHEMBL5537391 0.71 ALDH1A1 (0.33) ALDH1A1
SCHEMBL18381917 0.69
SCHEMBL20418887 0.68
SCHEMBL1016848 0.68
SCHEMBL3839581 0.67 ALDH1A1 (0.49) MEN1KMT2AALDH1A1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160134-A1 PREPARATION METHOD FOR AND CRYSTAL FORM OF 3-ARYLOXY-3-FIVE-MEMBERED HETEROARYL-PROPYLAMINE COMPOUND 漳州片仔癀药业股份有限公司 2021-08-19 WO disclosed
EP-3838900-A1 3-ARYLOXY-3-ARYL-PROPYLAMINE COMPOUND AND USES THEREOF Zhangzhou Pien Tze Huang Pharmaceutical Co., Ltd (CN) 2021-06-23 EP disclosed
WO-2020035070-A1 3-ARYLOXY-3-ARYL-PROPYLAMINE COMPOUND AND USES THEREOF 漳州片仔癀药业股份有限公司 2020-02-20 WO disclosed