SCHEMBL21744582

SCHEMBL21744582

CC(=O)c1cnc(-n2cccn2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.47
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 6/20 0.39
ALDH1A1 P00352 2/20 0.38
TP53 P04637 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CXCR4 P61073 1/20 0.37
HPGD P15428 2/20 0.37
MEN1 O00255 2/20 0.36
KAT6A Q92794 5/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
G6PD P11413 1/20 0.36
CYP2D6 P10635 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
JAK2 O60674 1/20 0.34
TYK2 P29597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3380687 0.88 LMNA (0.56) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL14910892 0.85 POLB (0.44) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL15351298 0.84 LMNA (0.48) LMNAKMT2AKDM4EALDH1A1TP53
SCHEMBL13822152 0.77 MAPT (0.37) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL29903403 0.77 MAPT (0.42) LMNAKMT2AKDM4EALDH1A1MEN1
SCHEMBL15072062 0.77 GRM4 (0.35) LMNAKMT2AKDM4EALDH1A1MEN1
SCHEMBL3377817 0.74 ADORA2A (0.41) LMNAKMT2AKDM4EALDH1A1MEN1
SCHEMBL14910553 0.74 LMNA (0.36) LMNAKMT2AKDM4EALDH1A1RXFP1
SCHEMBL24921598 0.74 KDM4E (0.38) KMT2AKDM4EALDH1A1HPGDMEN1
SCHEMBL10161002 0.74 MAPT (0.36) LMNAKMT2AKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035065-A1 PYRAZOLE DERIVATIVE AS RET INHIBITOR 南京明德新药研发有限公司 2020-02-20 WO disclosed