SCHEMBL21744943

SCHEMBL21744943

Cc1cc(NC2=NNC(C)C2)nc(N2CCNCC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.40
BPTF Q12830 2/20 0.38
KARS1 Q15046 2/20 0.37
CASP1 P29466 1/20 0.37
CASP4 P49662 1/20 0.37
CASP5 P51878 1/20 0.37
ROCK1 Q13464 2/20 0.36
ADRB1 P08588 1/20 0.36
NCF1 P14598 1/20 0.36
HRH4 Q9H3N8 2/20 0.36
AURKA O14965 2/20 0.34
RIPK1 Q13546 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
CHEK1 O14757 1/20 0.33
MAP3K12 Q12852 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18153318 0.75 BPTF (0.65) DPP4BPTFKARS1CASP1CASP4
Hydrochloric Acid SCHEMBL28463160 0.72 AURKA (0.55) DPP4AURKARIPK1CHEK1RET
SCHEMBL17303961 0.71 HRH4 (0.54) CASP1CASP4CASP5ROCK1ADRB1
SCHEMBL945117 0.68 CASP1 (0.53) CASP1CASP4CASP5ADRB1NCF1
SCHEMBL23299936 0.66 HRH4 (0.57) DPP4CASP1CASP4CASP5ADRB1
Hydrochloric Acid SCHEMBL15286713 0.65 CASP1 (0.49) CASP1CASP4CASP5ADRB1NCF1
SCHEMBL18278698 0.65 DPP4 (0.38) DPP4BPTFKARS1CASP1CASP4
SCHEMBL27389432 0.62 KDM4E (0.53) DPP4CASP1CASP4CASP5ADRB1
SCHEMBL16809209 0.61 NUDT1 (0.50) DPP4BPTFCASP1CASP4CASP5
SCHEMBL15286256 0.61 KDM4E (0.46) DPP4CASP1CASP4CASP5ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035065-A1 PYRAZOLE DERIVATIVE AS RET INHIBITOR 南京明德新药研发有限公司 2020-02-20 WO disclosed