SCHEMBL21752829

SCHEMBL21752829

Cc1onc(-c2ccccc2C(F)(F)F)c1CO

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NR1H4 Q96RI1 5/20 0.43
HSD11B1 P28845 2/20 0.42
GABRA5 P31644 4/20 0.42
NTRK1 P04629 1/20 0.41
P2RX7 Q99572 4/20 0.40
MAPT P10636 1/20 0.39
DPP4 P27487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27936768 0.84 NR1H4 (0.54) GPBAR1L3MBTL1NR1H4GABRA5NTRK1
SCHEMBL29384878 0.81 NR1H4 (0.57) NR1H4
SCHEMBL19202559 0.81 NR1H4 (0.57) NR1H4
SCHEMBL2929241 0.81 GABRA5 (0.49) GPBAR1L3MBTL1GABRA5MAPT
SCHEMBL30395460 0.76 GPBAR1 (0.63) GPBAR1L3MBTL1NTRK1MAPT
SCHEMBL12544227 0.76 GPBAR1 (0.63) GPBAR1L3MBTL1NTRK1MAPT
SCHEMBL2962082 0.75 GABRA5 (0.51) GPBAR1GABRA5P2RX7MAPT
SCHEMBL19033 0.75 HSD17B10 (0.65) GPBAR1L3MBTL1
SCHEMBL21752793 0.74 GPBAR1 (0.49) GPBAR1L3MBTL1NR1H4HSD11B1NTRK1
SCHEMBL21840049 0.74 NR1H4 (0.56) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020040343-A1 ISOXAZOLE DERIVATIVES AND PREPARATION PROCESS THEREOF IL-YANG PHARM. CO., LTD. (KR) 2020-02-27 WO disclosed