SCHEMBL21753046

SCHEMBL21753046

C=CCOC(=O)C(C)(C)Oc1c(C)cc(C=O)cc1C

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.40
FBP1 P09467 5/20 0.38
PPARA Q07869 12/20 0.36
PPARD Q03181 8/20 0.36
PPARG P37231 4/20 0.36
CYP3A4 P08684 2/20 0.34
ABCB11 O95342 1/20 0.34
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
HTR2A P28223 1/20 0.34
PMP22 Q01453 1/20 0.34
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL814693 0.86 FBP1 (0.49) SRCFBP1PPARAPPARDPPARG
SCHEMBL21758957 0.81 HPGD (0.33) FBP1PPARAPPARDPPARGCYP3A4
SCHEMBL20702486 0.80 SRC (0.46) SRCFBP1PPARAPPARDPPARG
SCHEMBL11893197 0.79 SRC (0.45) SRCFBP1PPARAPPARDPPARG
SCHEMBL5480699 0.78 FBP1 (0.46) SRCFBP1PPARAPPARDPPARG
SCHEMBL5479986 0.76 FBP1 (0.46) SRCFBP1PPARACYP3A4ABCB11
SCHEMBL5472116 0.76 PPARA (0.53) SRCPPARAPPARDPPARGKCNH2
SCHEMBL14290098 0.76 SRC (0.43) SRCFBP1PPARAPPARDPPARG
SCHEMBL21758868 0.76 PPARA (0.71) PPARAPPARDPPARG
SCHEMBL21188213 0.73 FBP1 (0.48) FBP1PPARAPPARDPPARGCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039297-A1 NOVEL COMPOUNDS AND THEIR USE IN PREPARATION OF ELAFIBRANOR AND PHARMACEUTICAL ACCEPTABLE SALTS THEREOF MANKIND PHARMA LTD. (IN) 2020-02-27 WO disclosed
WO-2020039297-A1 NOVEL COMPOUNDS AND THEIR USE IN PREPARATION OF ELAFIBRANOR AND PHARMACEUTICAL ACCEPTABLE SALTS THEREOF MANKIND PHARMA LTD. (IN) 2020-02-27 WO disclosed