SCHEMBL21753280

SCHEMBL21753280

N#Cc1ccc(N2CC3(CCN(C(=O)O)CC3)CC2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACA Q13085 8/20 0.56
ITGB3 P05106 7/20 0.51
ITGA2B P08514 7/20 0.51
KCNJ1 P48048 1/20 0.48
ACACB O00763 4/20 0.44
CYP2D6 P10635 1/20 0.44
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21753329 0.83 ACACA (0.53) ACACAITGB3ITGA2BKCNJ1ACACB
SCHEMBL16430910 0.80 ACACA (0.48) ACACAITGB3ITGA2BKCNJ1ACACB
SCHEMBL21753321 0.78 ITGB3 (0.48) ITGB3ITGA2BCYP2D6MEN1CYP1A2
SCHEMBL21753334 0.78 OPRL1 (0.58) ACACAITGB3ITGA2BCYP2D6
SCHEMBL6620291 0.77 SSTR5 (0.49)
SCHEMBL485114 0.76 AR (0.47) ITGB3ITGA2BCYP2D6MEN1CYP1A2
SCHEMBL17444273 0.74 OPRL1 (0.66) KCNJ1
SCHEMBL17444275 0.74 OPRL1 (0.66) KCNJ1
SCHEMBL16637299 0.73 POLB (0.45) ACACAKCNJ1CYP2D6TSHRPOLB
SCHEMBL29550707 0.71 TSHR (0.42) CYP2D6MEN1CYP1A2CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039029-A1 SPIRO COMPOUNDS AS GLYCOSIDASE INHIBITORS ASCENEURON S. A. (CH) 2020-02-27 WO disclosed