SCHEMBL21753313

SCHEMBL21753313

N#Cc1cnn(-c2ccc(CO)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.48
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
GCGR P47871 1/20 0.38
ACACB O00763 1/20 0.38
VHL P40337 1/20 0.37
ELOC Q15369 1/20 0.37
ELOB Q15370 1/20 0.37
CYP19A1 P11511 1/20 0.37
ALKBH1 Q13686 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
EGLN2 Q96KS0 1/20 0.35
GAA P10253 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1549833 0.84 NOTUM (0.55) NOTUMCYP11B1CYP11B2CYP19A1ALKBH1
SCHEMBL21753342 0.84 CYP19A1 (0.40) NOTUMCYP11B1CYP11B2GCGRACACB
SCHEMBL7259245 0.82 QPCT (0.45) GCGRACACBALKBH1EGLN1
SCHEMBL1682507 0.81 CA12 (0.47) NOTUMGCGRCYP19A1GAASCN9A
SCHEMBL28241532 0.78 MAOB (0.39) NOTUMCYP11B1CYP11B2GCGRCYP19A1
SCHEMBL2214866 0.78 GAA (0.53) ACACBGAA
SCHEMBL21525502 0.76 HPGDS (0.53) GCGR
SCHEMBL25365261 0.75 NOTUM (0.44) NOTUMGCGRVHLELOCELOB
SCHEMBL15729239 0.75 VHL (0.40) NOTUMGCGRVHLELOCELOB
SCHEMBL21753234 0.75 KMT2A (0.47) VHLELOCELOBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12016852-B2 Pyrrolidine glycosidase inhibitors ASCENEURON SA (CH) 2024-06-25 US disclosed
US-12016852-B2 Pyrrolidine glycosidase inhibitors ASCENEURON SA (CH) 2024-06-25 US disclosed
US-20210213005-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2021-07-15 US disclosed
US-20210213005-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2021-07-15 US disclosed
WO-2020039027-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON S. A. (CH) 2020-02-27 WO disclosed
WO-2020039027-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON S. A. (CH) 2020-02-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12016852-B2 Pyrrolidine glycosidase inhibitors PREP, GAA, DNPEP NOTUM 476/4885CYP11B1 2519/4885CYP11B2 2659/4885
US-20210213005-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS PREP, GAA, DNPEP NOTUM 358/4885CYP11B1 2625/4885CYP11B2 2834/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.