SCHEMBL21753522

SCHEMBL21753522

CCOC(=O)C(NN)C(=O)Cc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.46
KDM4E B2RXH2 4/20 0.44
EPHX2 P34913 1/20 0.43
PPARG P37231 1/20 0.43
POLB P06746 1/20 0.43
APEX1 P27695 1/20 0.43
RAB9A P51151 1/20 0.43
MAPT P10636 3/20 0.42
KMT2A Q03164 5/20 0.42
MEN1 O00255 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALDH1A1 P00352 2/20 0.42
GAA P10253 3/20 0.41
LMNA P02545 3/20 0.41
HTT P42858 1/20 0.41
KCNQ3 O43525 3/20 0.41
KCNQ2 O43526 3/20 0.41
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40
CCR6 P51684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653111 0.79 TDP1 (0.63) TDP1KDM4EEPHX2PPARGPOLB
SCHEMBL21753573 0.79 RAB9A (0.41) TDP1KDM4EEPHX2PPARGPOLB
SCHEMBL1287236 0.77 TDP1 (0.45) TDP1KDM4EEPHX2PPARGPOLB
SCHEMBL16144858 0.73 TDP1 (0.51) TDP1KDM4EPOLBAPEX1RAB9A
SCHEMBL1626240 0.73 TDP1 (0.54) TDP1KDM4EPPARGPOLBAPEX1
SCHEMBL3411918 0.72 CA12 (0.63) TDP1KDM4EMAPTKMT2AMEN1
SCHEMBL839736 0.71 PPARG (0.51) TDP1KDM4EEPHX2PPARGPOLB
SCHEMBL699965 0.71 KDM4E (0.50) TDP1KDM4EPOLBAPEX1RAB9A
SCHEMBL1064642 0.71 PPARG (0.51) TDP1KDM4EEPHX2PPARGPOLB
SCHEMBL838697 0.71 PPARG (0.51) TDP1KDM4EEPHX2PPARGPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020038460-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR 南京药捷安康生物科技有限公司 2020-02-27 WO disclosed