SCHEMBL21753531

SCHEMBL21753531

NC(=O)c1cn(Cc2ccccc2)ccc1=O

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
ADRA1D P25100 5/20 0.49
CYP2C19 P33261 1/20 0.49
PARP1 P09874 3/20 0.45
BRD4 O60885 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
CYP2D6 P10635 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
POLB P06746 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PARP2 Q9UGN5 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11557346 0.87 CA12 (0.55) CA12CA1CA2CA9CYP2C19
SCHEMBL4155873 0.79 CYP2C19 (0.53) CA12CA1CA2CA9ADRA1D
SCHEMBL10314669 0.79 TSHR (0.53) CA12CA1CA2CA9KDM4E
SCHEMBL15333147 0.74 NPC1 (0.45) CA12CA1CA2CA9CYP2C19
SCHEMBL28856280 0.73 CA12 (0.38) CA12CA1CA2CA9KMT2A
SCHEMBL21776615 0.73 CCNC (0.58) ADRA1DPARP1BRD4KDM4E
SCHEMBL353268 0.72 NOTUM (0.51) CYP2C19KMT2APOLB
Hydrochloric Acid SCHEMBL28856209 0.72 CA12 (0.37) CA12CA1CA2CA9KMT2A
SCHEMBL28771070 0.71 LMNA (0.58) CYP2C19
SCHEMBL2514239 0.71 CYP2C19 (0.55) CA12CA1CA2CA9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020038460-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR 南京药捷安康生物科技有限公司 2020-02-27 WO disclosed