SCHEMBL28856280

SCHEMBL28856280

NC(=O)c1cn(CC(F)(F)F)ccc1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.38
CA1 P00915 5/20 0.38
CA2 P00918 5/20 0.38
CA9 Q16790 5/20 0.38
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TYR P14679 1/20 0.35
DOHH Q9BU89 1/20 0.35
LMNA P02545 2/20 0.33
XBP1 P17861 2/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CDC7 O00311 1/20 0.32
METAP2 P50579 2/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28856209 0.98 CA12 (0.37) CA12CA1CA2CA9KDM4E
SCHEMBL28842741 0.78 AKR1B1 (0.38) CA12CA1CA2CA9ALDH1A1
SCHEMBL12949753 0.76 TYR (0.49) CA12CA1CA2CA9KDM4E
SCHEMBL21753531 0.73 CA12 (0.56) CA12CA1CA2CA9KDM4E
SCHEMBL13555516 0.73 NR3C1 (0.33) CA12CA1CA2CA9
SCHEMBL29812137 0.70 AXL (0.53) CA12CA1CA2CA9KDM4E
SCHEMBL715572 0.68 CA12 (0.47) CA12CA1CA2CA9KDM4E
SCHEMBL31069484 0.66 KMT2A (0.42) CA12CA1CA2CA9KDM4E
SCHEMBL29811977 0.65 IRAK4 (0.35) CA12CA1CA2CA9KDM4E
SCHEMBL22245577 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104185627-B Pyridone Derivatives 第三共株式会社 2018-01-12 CN disclosed