SCHEMBL21753620

SCHEMBL21753620

CC(=O)Nc1ccc(N2CCN(C)CC2)cc1[N+](=O)[O-]

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.61
SIRT6 Q8N6T7 10/20 0.60
MAPK1 P28482 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
HTR6 P50406 5/20 0.55
NPSR1 Q6W5P4 1/20 0.53
ALDH1A1 P00352 1/20 0.53
KDM4E B2RXH2 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL975415 0.90 MAPT (0.59) MAPTMAPK1L3MBTL1NPSR1ALDH1A1
SCHEMBL16262967 0.88 MAPT (0.51) MAPTSIRT6NPSR1ALDH1A1KDM4E
SCHEMBL16262970 0.88 MAPT (0.51) MAPTSIRT6NPSR1ALDH1A1KDM4E
SCHEMBL5457891 0.86 MAPT (0.64) MAPTMAPK1NPSR1ALDH1A1
SCHEMBL19633486 0.85 KMT2A (0.50) MAPTSIRT6MAPK1NPSR1ALDH1A1
SCHEMBL19633305 0.82 MAPT (0.54) MAPTMAPK1NPSR1ALDH1A1
SCHEMBL16270618 0.82 MAPT (0.61) MAPTSIRT6NPSR1ALDH1A1KDM4E
SCHEMBL5332939 0.81 ALDH1A1 (0.48) MAPTSIRT6MAPK1L3MBTL1ALDH1A1
SCHEMBL19633404 0.81 MAPT (0.53) MAPTMAPK1NPSR1ALDH1A1
SCHEMBL14669416 0.81 ALDH1A1 (0.48) MAPTSIRT6MAPK1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110857300-B Condensed ring triazole compounds, preparation method and application 上海凌达生物医药有限公司 2021-11-05 CN disclosed
CN-109721600-B Nitrogen-containing fused ring compounds and preparation method and application thereof 上海凌达生物医药有限公司 2021-04-27 CN disclosed
CN-110857300-A Condensed ring triazole compounds, preparation method and application 如东凌达生物医药科技有限公司 2020-03-03 CN disclosed
WO-2020038458-A1 CLASS OF FUSED RING TRIAZOLE COMPOUND, PREPARATION METHOD, AND USE 如东凌达生物医药科技有限公司 2020-02-27 WO disclosed