SCHEMBL2175629

SCHEMBL2175629

CCC(C)N(NNCc1ccc(-c2ccccn2)cc1)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.45
EPHX1 P07099 1/20 0.42
CYP2D6 P10635 1/20 0.42
EPHX2 P34913 1/20 0.42
HPGDS O60760 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
CCNE1 P24864 7/20 0.41
CDK2 P24941 7/20 0.41
CDK5 Q00535 4/20 0.41
CCNK O75909 2/20 0.39
CDK9 P50750 2/20 0.39
CDK12 Q9NYV4 2/20 0.39
DYRK1A Q13627 2/20 0.39
PPARG P37231 1/20 0.39
CCNT1 O60563 1/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNA2 P20248 1/20 0.39
CCND1 P24385 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179440 0.77 HDAC3 (0.49) SLC6A9HPGD
SCHEMBL3550411 0.77 HCAR2 (0.41) SLC6A9EPHX1CYP2D6EPHX2HPGDS
SCHEMBL893594 0.75 HCAR2 (0.55) EPHX1CYP2D6EPHX2HPGDSHCAR2
SCHEMBL3804430 0.73 DPP4 (0.45) SLC6A9HCAR2PPARG
SCHEMBL2175634 0.73 EPHX1 (0.42) EPHX1CYP2D6EPHX2HPGDSHCAR2
SCHEMBL2773101 0.72 HPGDS (0.56) EPHX1CYP2D6EPHX2HPGDSHCAR2
SCHEMBL3550406 0.72 HCAR2 (0.43) EPHX1CYP2D6EPHX2HCAR2CCNE1
SCHEMBL7911949 0.72 HCAR2 (0.46) EPHX1CYP2D6EPHX2HPGDSHCAR2
SCHEMBL13315147 0.72 CYP2D6 (0.47) EPHX1CYP2D6EPHX2HCAR2CCNE1
SCHEMBL7716958 0.71 EPHX1 (0.44) EPHX1CYP2D6EPHX2HPGDSHCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080562-A1 NOVEL AZA-PEPTIDES CONTAINING 2,2-DISUBSTITUTED CYCLOBUTYL AND/OR SUBSTITUTED ALKOXY BENZYL DERIVATIVES AS ANTIVIRALS HETERO RESEARCH FOUNDATION (IN) 2011-07-07 WO disclosed