SCHEMBL2175634

SCHEMBL2175634

CC(CCNNCc1ccc(-c2ccccn2)cc1)NC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.42
CYP2D6 P10635 1/20 0.42
EPHX2 P34913 1/20 0.42
HCAR2 Q8TDS4 1/20 0.41
CDK2 P24941 9/20 0.41
CCNE1 P24864 8/20 0.41
CDK5 Q00535 5/20 0.41
CHRM4 P08173 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
KLKB1 P03952 1/20 0.39
CCNT1 O60563 1/20 0.39
CCNA2 P20248 1/20 0.39
CSNK1A1 P48729 1/20 0.39
CDK9 P50750 1/20 0.39
CCNA1 P78396 1/20 0.39
DYRK1A Q13627 1/20 0.39
CDK5R1 Q15078 1/20 0.39
HPGDS O60760 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179773 0.83 CDK2 (0.46) CDK2CCNE1CDK5CCNT1CCNA2
SCHEMBL3550406 0.79 HCAR2 (0.43) EPHX1CYP2D6EPHX2HCAR2CDK2
SCHEMBL893594 0.78 HCAR2 (0.55) EPHX1CYP2D6EPHX2HCAR2CHRM4
SCHEMBL2179441 0.77 HDAC3 (0.49) SMN1; SMN2
SCHEMBL3558719 0.76 UGT1A1 (0.47) EPHX1CYP2D6EPHX2HCAR2CDK2
SCHEMBL2773101 0.75 HPGDS (0.56) EPHX1CYP2D6EPHX2HCAR2CHRM4
SCHEMBL2175629 0.73 SLC6A9 (0.45) EPHX1CYP2D6EPHX2HCAR2CDK2
SCHEMBL7911949 0.72 HCAR2 (0.46) EPHX1CYP2D6EPHX2HCAR2CDK2
SCHEMBL13315147 0.72 CYP2D6 (0.47) EPHX1CYP2D6EPHX2HCAR2CDK2
SCHEMBL4252334 0.71 MME (0.48) CYP2D6HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080562-A1 NOVEL AZA-PEPTIDES CONTAINING 2,2-DISUBSTITUTED CYCLOBUTYL AND/OR SUBSTITUTED ALKOXY BENZYL DERIVATIVES AS ANTIVIRALS HETERO RESEARCH FOUNDATION (IN) 2011-07-07 WO disclosed