SCHEMBL21756928

SCHEMBL21756928

CCc1ccc(I)cc1CNC

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 15/20 0.39
HTR2A P28223 7/20 0.39
KCNH2 Q12809 7/20 0.39
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SLC6A2 P23975 8/20 0.35
SLC6A3 Q01959 5/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104506 0.83 IDO1 (0.36) SLC6A4SLC6A2
SCHEMBL22765684 0.79 KDM4E (0.49) SLC6A4HTR2AKCNH2KDM4EALDH1A1
SCHEMBL31378001 0.76 SLC6A4 (0.36) SLC6A4HTR2AKCNH2SLC6A2SLC6A3
SCHEMBL8145201 0.76 SLC6A4 (0.56) SLC6A4HTR2AKCNH2SLC6A2SLC6A3
SCHEMBL16831106 0.75 SLC6A4 (0.42) SLC6A4SLC6A2
SCHEMBL24422626 0.74 KDM4E (0.38) SLC6A4HTR2AKCNH2KDM4EALDH1A1
SCHEMBL18619507 0.73 TNIK (0.38) SLC6A4KCNH2KDM4EALDH1A1SLC6A2
SCHEMBL28543732 0.73 IDO1 (0.35) SLC6A4SLC6A2
SCHEMBL13761530 0.73 APP (0.35) SLC6A4SLC6A2
SCHEMBL21756948 0.73 SLC6A2 (0.38) SLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-9403829-B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use SIGNAL PHARMACEUTICALS, LLC (US) 2016-08-02 US disclosed