SCHEMBL21756941

SCHEMBL21756941

Nc1ccc(Oc2ccc(C3CC3)cc2)c(N)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.45
ALDH1A1 P00352 5/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
KDM4E B2RXH2 2/20 0.45
CYP2D6 P10635 1/20 0.45
HPGD P15428 1/20 0.45
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CYP3A4 P08684 2/20 0.40
SCN5A Q14524 2/20 0.39
SCN9A Q15858 2/20 0.39
KCNH2 Q12809 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10049050 0.93 ESR2 (0.44) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL12220514 0.93 ESR2 (0.42) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL5682640 0.92 HAO1 (0.43) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL10033588 0.90 SMN1; SMN2 (0.38) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL21765332 0.90 MAPT (0.45) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL10017553 0.89 SLC6A4 (0.41) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL17720303 0.89 ESR2 (0.40) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL17722779 0.89 MAPT (0.37) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL16171980 0.87 CYP2C9 (0.47) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL13910064 0.87 SLC6A2 (0.40) MAPTALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-9403829-B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use SIGNAL PHARMACEUTICALS, LLC (US) 2016-08-02 US disclosed