SCHEMBL2175697

SCHEMBL2175697

CC(=O)N1CCCC1C(=O)Nc1ccc(-c2nnc(-c3ccc(NC(=O)C4CCCN4C(=O)Cc4ccccc4)cc3)o2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
HCRTR1 O43613 2/20 0.49
HCRTR2 O43614 2/20 0.49
KDM4E B2RXH2 4/20 0.48
HSD17B10 Q99714 4/20 0.48
LMNA P02545 2/20 0.48
MEN1 O00255 2/20 0.48
HPGD P15428 2/20 0.48
KMT2A Q03164 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ITGB1 P05556 4/20 0.47
ITGA4 P13612 4/20 0.47
KCNH2 Q12809 1/20 0.47
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
MAPT P10636 1/20 0.46
MAPK10 P53779 1/20 0.45
CACNA1B Q00975 1/20 0.45
APBA1 Q02410 1/20 0.45
CPA1 P15085 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12489099 1.00 ALDH1A1 (0.50) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL2193840 0.95 HSD17B10 (0.53) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL2195941 0.95 HSD17B10 (0.53) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL12488545 0.90 ALDH1A1 (0.42) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL2179845 0.90 ALDH1A1 (0.42) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL2190466 0.89 HCRTR1 (0.47) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL2194705 0.89 HCRTR1 (0.47) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL2194905 0.88 ALDH1A1 (0.51) ALDH1A1KDM4EHSD17B10LMNAMEN1
SCHEMBL2179610 0.86 ALDH1A1 (0.52) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10
SCHEMBL12488611 0.86 ALDH1A1 (0.52) ALDH1A1HCRTR1HCRTR2KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011082077-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-07-07 WO claimed