SCHEMBL21759876

SCHEMBL21759876

CN(C)c1ccc(C(=O)c2nc3ccccc3[nH]2)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCND3 P30281 1/20 0.56
CDK6 Q00534 1/20 0.56
CNR2 P34972 1/20 0.55
RAB9A P51151 4/20 0.53
NPC1 O15118 3/20 0.53
HPGD P15428 2/20 0.53
PDE10A Q9Y233 9/20 0.51
MAPT P10636 2/20 0.50
ALDH1A1 P00352 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7199487 0.88 CCND3 (0.69) CCND3CDK6RAB9ANPC1HPGD
SCHEMBL13042221 0.84 MAPT (0.60) CCND3CDK6RAB9ANPC1HPGD
SCHEMBL3966827 0.83 CCND3 (0.67) CCND3CDK6RAB9ANPC1HPGD
SCHEMBL1303899 0.82 CCND3 (0.61) CCND3CDK6RAB9ANPC1HPGD
SCHEMBL250171 0.79 CCND3 (0.70) CCND3CDK6RAB9ANPC1HPGD
SCHEMBL9373255 0.79 CCND3 (0.61) CCND3CDK6RAB9ANPC1PDE10A
Hydrochloric Acid SCHEMBL7000982 0.78 CCND3 (0.68) CCND3CDK6RAB9ANPC1HPGD
SCHEMBL8350123 0.78 CCND3 (0.60) CCND3CDK6RAB9ANPC1HPGD
SCHEMBL14804457 0.76 PDE10A (0.72) PDE10A
SCHEMBL10428595 0.74 PDE10A (0.53) CCND3CDK6RAB9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585462-B1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICALS CO (JP) 2020-02-26 EP disclosed