SCHEMBL21763371

SCHEMBL21763371

CN1CCN(c2ncc(-c3ccc4c(C=O)cccc4c3)s2)CC1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.49
ERN1 O75460 3/20 0.41
KCNH2 Q12809 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
MET P08581 1/20 0.39
HDAC2 Q92769 1/20 0.38
TNKS O95271 2/20 0.38
TP53 P04637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ESR2 Q92731 1/20 0.38
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
KIT P10721 1/20 0.36
KDR P35968 1/20 0.36
FLT3 P36888 1/20 0.36
WNT1 P04628 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12675652 0.82 ERN1 (0.62) TDP1ERN1
SCHEMBL21763575 0.80 SMN1; SMN2 (0.49) ERN1ALDH1A1MAPTTP53POLB
SCHEMBL27891120 0.75 TDP1 (0.53) TDP1ALDH1A1MAPTMETHDAC2
SCHEMBL21763659 0.74 HTR3A (0.56) ERN1ALDH1A1
SCHEMBL21763657 0.73 ERN1 (0.49) ERN1KCNH2KDRWNT1GSK3B
SCHEMBL8249743 0.71 CHEK1 (0.53) TDP1KCNH2HDAC2TP53NPSR1
SCHEMBL21763595 0.71 ERN1 (0.60) ERN1KCNH2ALDH1A1MAPT
SCHEMBL21763695 0.70 ERN1 (0.54) ERN1KCNH2TNKS
SCHEMBL444649 0.70 TDP1 (0.50) TDP1KCNH2ALDH1A1HDAC2TP53
SCHEMBL1554083 0.68 TDP1 (1.00) TDP1ALDH1A1MAPTHDAC2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496230-B1 IRE-1 ALPHA INHIBITORS FOSUN ORINOVE PHARMATECH INC (CN) 2020-02-26 EP disclosed