SCHEMBL21763580

SCHEMBL21763580

CN1CCN(C(=O)c2ccc(Oc3ccc4c(C=O)cccc4c3)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.51
TSHR P16473 1/20 0.51
ERN1 O75460 4/20 0.48
NPC1 O15118 1/20 0.47
SCN9A Q15858 1/20 0.45
POLB P06746 2/20 0.44
APP P05067 1/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
GAA P10253 2/20 0.42
SCN7A Q01118 1/20 0.42
KCNH2 Q12809 1/20 0.42
MAPT P10636 2/20 0.42
CRHBP P24387 1/20 0.42
HTT P42858 1/20 0.42
CRHR2 Q13324 1/20 0.42
BTK Q06187 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12675810 0.82 ERN1 (0.65) HPGDTSHRERN1NPC1SCN9A
SCHEMBL21763595 0.76 ERN1 (0.60) HPGDTSHRERN1KCNH2MAPT
SCHEMBL13551886 0.75 HPGD (0.47) HPGDTSHRERN1NPC1SCN9A
SCHEMBL21763695 0.73 ERN1 (0.54) ERN1NPC1KCNH2KDM4ESMN1; SMN2
SCHEMBL21763560 0.72 ERN1 (0.70) ERN1NPC1MAPT
SCHEMBL24368722 0.72 HPGD (0.54) HPGDTSHRSCN9AMEN1KMT2A
SCHEMBL21763684 0.71 KDM4E (0.41) HPGDTSHRERN1NPC1MAPT
SCHEMBL21763657 0.70 ERN1 (0.49) ERN1NPC1KMT2AKCNH2KDM4E
SCHEMBL21763659 0.70 HTR3A (0.56) ERN1NPC1MEN1CYP1A2KMT2A
SCHEMBL10724841 0.69 POLB (0.81) HPGDTSHRNPC1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496230-B1 IRE-1 ALPHA INHIBITORS FOSUN ORINOVE PHARMATECH INC (CN) 2020-02-26 EP disclosed