SCHEMBL21763899

SCHEMBL21763899

O=C(Nc1ccc2ncccc2c1)c1cccc(-c2nnc(SCC(O)O)[nH]2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.52
RAB9A P51151 6/20 0.52
CASP3 P42574 1/20 0.52
SENP8 Q96LD8 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
SENP6 Q9GZR1 1/20 0.52
PABPC1 P11940 1/20 0.52
POLB P06746 2/20 0.47
PARP1 P09874 1/20 0.44
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
BRAF P15056 1/20 0.42
MMP9 P14780 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17213024 0.90 PABPC1 (0.55) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL18540543 0.90 NPC1 (0.52) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL17213099 0.73 NPC1 (0.51) NPC1RAB9APOLBPARP1ALDH1A1
SCHEMBL17213001 0.73 RAB9A (0.46) NPC1RAB9APOLBALDH1A1KMT2A
SCHEMBL17212996 0.72 SIRT2 (0.52) NPC1RAB9APOLBALDH1A1MAPT
SCHEMBL17213100 0.72 NR1H4 (0.48) NPC1RAB9APOLBALDH1A1MAPT
SCHEMBL18540510 0.72 KMT2A (0.53) NPC1RAB9APOLBALDH1A1MAPT
SCHEMBL18540535 0.71 SMN1; SMN2 (0.49) NPC1RAB9APOLBALDH1A1MAPT
SCHEMBL17213061 0.71 NPC1 (0.50) NPC1RAB9APOLBALDH1A1MAPT
SCHEMBL17212991 0.71 GRK6 (0.44) NPC1RAB9APOLBPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3134390-B1 SMALL MOLECULE INHIBITORS OF G PROTEIN COUPLED RECEPTOR 6 KINASE POLYPEPTIDES MAYO FOUND MEDICAL EDUCATION & RES (US) 2020-02-26 EP disclosed