SCHEMBL21768249

SCHEMBL21768249

COC(=O)[C@H]1CCN(CCCC(=O)O)[C@@H](C(F)(F)F)C1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
GAA P10253 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 2/20 0.33
LTA4H P09960 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP1A2 P05177 1/20 0.32
MAPK1 P28482 1/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.31
FKBP1A P62942 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21782043 1.00 ALDH1A1 (0.37) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL21768206 1.00 ALDH1A1 (0.37) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL22068089 0.82 GAA (0.40) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL23726895 0.79 SMN1; SMN2 (0.38) ALDH1A1GAASMN1; SMN2TP53MAPT
SCHEMBL21781967 0.79 ALDH1A1 (0.30) ALDH1A1SMN1; SMN2
SCHEMBL29939188 0.78 SMN1; SMN2 (0.38) ALDH1A1GAASMN1; SMN2TP53MAPT
SCHEMBL26544376 0.78 SMN1; SMN2 (0.38) ALDH1A1GAASMN1; SMN2TP53MAPT
SCHEMBL17802980 0.77 SMN1; SMN2 (0.43) ALDH1A1GAASMN1; SMN2TP53MAPT
SCHEMBL21781802 0.74 OPRD1 (0.30)
SCHEMBL8140913 0.72 SMN1; SMN2 (0.42) ALDH1A1GAANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110312730-B Cytotoxins and conjugates, uses thereof and methods of preparation 四川科伦博泰生物医药股份有限公司 2024-06-18 CN disclosed
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed